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SB-277011 hydrochloride

Glpbio
Catalog No:GC60334-10mM (in 1mL DMSO) CAS No.:215804-67-4 MDLNo:C28H31ClN4O Brand:Glpbio purity: 特性: Purpose:SB-277011hydrochloride(SB-277011Ahydrochloride)是一种强效、选择性、口服生物利用度和脑透多巴胺D3受体(D3R)拮抗剂,其Ki值在啮齿动物和人D3R分别为10.7nM和11.2nM。SB-277011hydrochloride对D3受体比其他多巴胺受体表现出80-100倍的选择性,,对D3,D2,5-HT1B 和5-HT1D受体的 pKi值分别为8.0,6.0,<5.2和5.9。DMSO: 50 mg/mL (105.26 mM; Need ultrasonic); H2O: 16.67 mg/mL (35.09 mM; Need ultrasonic)
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Product Overview
Product Name SB-277011 hydrochloride
CAS215804-67-4
MW475.02
MDLC28H31ClN4O
Storage conditionPowder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
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